Aspirin Tables:

Pharmacokinetics

Bioavailability Peak plasma level Plasma half-life Active metabolites Elimination
minimal variability 50% 30 minutes 20 minutes salicylic acid renal
All indications refer to quickly absorbed, unhydrolized aspirin. The latter is quickly metabolized (in part presystemically) to salicylic acid. Salicylic acid reaches peak plasma level in 1 to 2 hours, it has a dose dependent half-life (2-30 hours), and is partially eliminated hepatically.

Dose
Indication Administration
Initial loading dose
Dose Interval
Maintenance dose
Dose Interval
headache oral 500 mg 4 to 6 hours - -
platelet inhibition* oral 100 mg 24 hours 100 mg 24 hours
*The "ideal" dose is not known. For coronary heart disease 100 mg/day or less suffice; for other angiopathies higher doses (300-500 mg/day) have often been administered.

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